1003877-55-1
1003877-55-1
Chemical Structure
GSK-1562590
- CAS No.: 1003877-55-1
- Formula:C30H30Cl2N4O4
- Molecular Weight:581.49
InChIKey: QDUMEBKFKOODFN-SANMLTNESA-N
SMILES: NC(C1=CC=CC(C(C=C2)=CC=C2[C@H](CN3CCCC3)N(C)C(CN4C5=CC(Cl)=C(Cl)C=C5OCC4=O)=O)=C1)=O
Biological Activity: GSK-1562590 is a uropeptide-II receptor antagonist with high affinity and selectivity. GSK-1562590 exhibits significant antagonistic activity in multiple bioassays and, in contrast, displays relatively sustained receptor binding times. GSK-1562590 can inhibit human urinary peptide-II-induced aortic contraction in rats in experiments, and its effect can last for at least 24 hours[1].
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GSK-1562590 | GSK-1562590 is a uropeptide-II receptor antagonist with high affinity and selectivity. GSK-1562590 exhibits significant antagonistic activity in multiple bioassays and, in contrast, displays relatively sustained receptor binding times. GSK-1562590 can inhibit human urinary peptide-II-induced aortic contraction in rats in experiments, and its effect can last for at least 24 hours. | |||||||||||||||||||||
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