100678-32-8
Chemical Structure
Cibenzoline succinate
Synonym(s): Cifenline succinate; Ro 22-7796 succinate
- CAS No.: 100678-32-8
- Formula:C22H24N2O4
- Molecular Weight:380.44
IUPAC Name: 2-(2,2-diphenylcyclopropyl)-4,5-dihydro-1H-imidazole succinate
InChIKey: XFUIOIWYMHEPIE-UHFFFAOYSA-N
SMILES: O=C(O)CCC(O)=O.C1(C2C(C3=CC=CC=C3)(C4=CC=CC=C4)C2)=NCCN1
Biological Activity: Cibenzoline succinate (Cifenline succinate) is the succinate form of Cibenzoline (HY-106577). Cibenzoline succinate is an inhibitor for ATP-sensitive potassium (KATP) channel by affecting the pore-forming Kir6.2 subunit with IC50 of 22.2 µM. Cibenzoline succinate affects insulin secretion and exhibits antiarrhythmic and antidiabetic activities[1].
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Cibenzoline succinate | Cibenzoline succinate (Cifenline succinate) is the succinate form of Cibenzoline (HY-106577). Cibenzoline succinate is an inhibitor for ATP-sensitive potassium (KATP) channel by affecting the pore-forming Kir6.2 subunit with IC50 of 22.2 µM. Cibenzoline succinate affects insulin secretion and exhibits antiarrhythmic and antidiabetic activities. | |||||||||||||||||||||
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