103926-82-5
103926-82-5
Chemical Structure
Sepimostat dimethanesulfonate
Synonym(s): FUT-187
- CAS No.: 103926-82-5
- Formula:C23H27N5O8S2
- Molecular Weight:565.62
IUPAC Name: 6-carbamimidoylnaphthalen-2-yl 4-((4,5-dihydro-1H-imidazol-2-yl)amino)benzoate dimethanesulfonate
InChIKey: ICYICMXERRTCPY-UHFFFAOYSA-N
SMILES: O=C(OC1=CC=C2C=C(C(N)=N)C=CC2=C1)C3=CC=C(NC4=NCCN4)C=C3.CS(=O)(O)=O.CS(=O)(O)=O
Biological Activity: Sepimostat dimethanesulfonate (FUT-187) exhibits neuroprotective activity via NR2B N-methyl-D-aspartate receptor antagonism at the Ifenprodil-binding site of the NR2B subunit. Sepimostat dimethanesulfonate inhibits the Ifenprodil binding with a Ki value of 27.7 µM[1].
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Sepimostat dimethanesulfonate | Sepimostat dimethanesulfonate (FUT-187) exhibits neuroprotective activity via NR2B N-methyl-D-aspartate receptor antagonism at the Ifenprodil-binding site of the NR2B subunit. Sepimostat dimethanesulfonate inhibits the Ifenprodil binding with a Ki value of 27.7 µM. | |||||||||||||||||||||
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