1068515-53-6
1068515-53-6
Chemical Structure
KDM4-IN-3
- CAS No.: 1068515-53-6
- Formula:C17H14N4O
- Molecular Weight:290.32
IUPAC Name: 1-(1H-benzo[d]imidazol-2-yl)-3-methyl-4-phenyl-1H-pyrazol-5-ol
InChIKey: MGIRLDYHTMQKEV-UHFFFAOYSA-N
SMILES: OC1=C(C2=CC=CC=C2)C(C)=NN1C3=NC4=CC=CC=C4N3
Biological Activity: KDM4-IN-3 (Compound 15) is a KDM4 inhibitor (IC50 = 871 nM) that exhibits improved potency in biochemical assays. KDM4-IN-3 is cell-permeable and kills prostate cancer cells at low micro molar concentrations. KDM4-IN-3 inhibits growth of prostate cancer cell lines and increases the H3K9me3 abundance. KDM4-IN-3 can be studied in research for prostate cancer[1].
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KDM4-IN-3 | 99.36% | KDM4-IN-3 (Compound 15) is a KDM4 inhibitor (IC50 = 871 nM) that exhibits improved potency in biochemical assays. KDM4-IN-3 is cell-permeable and kills prostate cancer cells at low micro molar concentrations. KDM4-IN-3 inhibits growth of prostate cancer cell lines and increases the H3K9me3 abundance. KDM4-IN-3 can be studied in research for prostate cancer. | ||||||||||||||||||||
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