120770-34-5
120770-34-5
Chemical Structure
Draflazine
Synonym(s): R-75231; R88021
- CAS No.: 120770-34-5
- Formula:C30H33Cl2F2N5O2
- Molecular Weight:604.52
IUPAC Name: 1-(2-((4-amino-2,6-dichlorophenyl)amino)-2-oxoethyl)-4-(5,5-bis(4-fluorophenyl)pentyl)piperazine-2-carboxamide
InChIKey: IWMYIWLIESDFRZ-UHFFFAOYSA-N
SMILES: O=C(NC1=C(Cl)C=C(N)C=C1Cl)CN2C(C(N)=O)CN(CCCCC(C3=CC=C(F)C=C3)C4=CC=C(F)C=C4)CC2
Biological Activity: Draflazine (R-75231) is a ENT1 inhibitor. Draflazine (R-75231) completely reverses the hypersensitivity in the complete Freund’s adjuvant (CFA) model of mechanical hyperalgesia and the carrageenan inflammation model of thermal and mechanical hyperalgesia[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Draflazine | 99.06% | Draflazine (R-75231) is a ENT1 inhibitor. Draflazine (R-75231) completely reverses the hypersensitivity in the complete Freund’s adjuvant (CFA) model of mechanical hyperalgesia and the carrageenan inflammation model of thermal and mechanical hyperalgesia. | ||||||||||||||||||||
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