1216074-15-5
1216074-15-5
Chemical Structure
5-HT2CR agonist 1
- CAS No.: 1216074-15-5
- Formula:C13H14ClNO
- Molecular Weight:235.71
InChIKey: OSLHZPLWTXHOAZ-UHFFFAOYSA-N
SMILES: ClC1=CC=C2C=CC3(OC2=C1)CCNCC3
Biological Activity: 5-HT2CR agonist 1 (compound 8), a 7-chloro analogue, is a selective 5-HT2CR partial agonist (Emax=71.09%) with an EC50 value of 121.5 nM and no observed activity toward 5-HT2AR or 5-HT2BR. 5-HT2CR agonist 1 exhibits no recruitment activity for β-arrestin and shows low inhibition of hERG at 10 μM[1].
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5-HT2CR agonist 1 | 5-HT2CR agonist 1 (compound 8), a 7-chloro analogue, is a selective 5-HT2CR partial agonist (Emax=71.09%) with an EC50 value of 121.5 nM and no observed activity toward 5-HT2AR or 5-HT2BR. 5-HT2CR agonist 1 exhibits no recruitment activity for β-arrestin and shows low inhibition of hERG at 10 μM. | |||||||||||||||||||||
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