1228817-38-6
1228817-38-6
Chemical Structure
Mps1-IN-2
- CAS No.: 1228817-38-6
- Formula:C26H36N6O3
- Molecular Weight:480.60
IUPAC Name: 9-cyclopentyl-2-((2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl)amino)-5-methyl-5,7,8,9-tetrahydro-6H-pyrimido[4,5-b][1,4]diazepin-6-one
InChIKey: WELBJLUKWAJOQV-UHFFFAOYSA-N
SMILES: CN(C1=CN=C(NC2=C(OCC)C=C(N3CCC(O)CC3)C=C2)N=C1N(C4CCCC4)CC5)C5=O
Biological Activity: Mps1-IN-2 is a potent, selective and ATP-competitive dual Mps1/Plk1 inhibitor, with an IC50 and a Kd of 145 nM and 12 nM for Mps1 and a Kd of 61 nM for Plk1.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Mps1-IN-2 | 98.08% | Mps1-IN-2 is a potent, selective and ATP-competitive dual Mps1/Plk1 inhibitor, with an IC50 and a Kd of 145 nM and 12 nM for Mps1 and a Kd of 61 nM for Plk1. | ||||||||||||||||||||
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