1234479-76-5
1234479-76-5
Chemical Structure
ERK5-IN-1
- CAS No.: 1234479-76-5
- Formula:C25H29N7O2
- Molecular Weight:459.54
IUPAC Name: 2-((2-methoxy-4-(4-methylpiperazin-1-yl)phenyl)amino)-5,11-dimethyl-5,11-dihydro-6H-benzo[e]pyrimido[5,4-b][1,4]diazepin-6-one
InChIKey: DDTPGANIPBKTNU-UHFFFAOYSA-N
SMILES: O=C1C2=C(C=CC=C2)N(C)C3=NC(NC4=C(OC)C=C(N5CCN(C)CC5)C=C4)=NC=C3N1C
Biological Activity: ERK5-IN-1 is a potent ERK5 inhibitor with an IC50 of 87±7 nM. ERK5-IN-1 also inhibits LRRK2[G2019S] with an IC50 of 26 nM.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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ERK5-IN-1 | 99.55% | ERK5-IN-1 is a potent ERK5 inhibitor with an IC50 of 87±7 nM. ERK5-IN-1 also inhibits LRRK2[G2019S] with an IC50 of 26 nM. | ||||||||||||||||||||
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