1312799-06-6
1312799-06-6
Chemical Structure
FFA2 agonist-1
- CAS No.: 1312799-06-6
- Formula:C25H22ClNO4
- Molecular Weight:435.90
SMILES: O=C(C1=CC=C(C2=C(C=CC=C2)OC)C=C1)N3[C@@H](C4=C(C=CC=C4)Cl)CC[C@H]3C(O)=O
Biological Activity: FFA2 agonist-1 (Compound 4) is the agonist for Free fatty acid receptor 2 (FFA2/GPR43) with an EC50 of 81 nM. FFA2 agonist-1 exhibits activity in β-arrestin-2 recruitment assay and cAMP inhibition assay with EC50 of 1.2 μM and 0.53 μM. FFA2 agonist-1 leads to appetite regulating peptide YY (PYY) mucosal responses, inhibits the fat accumulation, intestinal functions and food intake, and can be used for obesity research[1].
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FFA2 agonist-1 | FFA2 agonist-1 (Compound 4) is the agonist for Free fatty acid receptor 2 (FFA2/GPR43) with an EC50 of 81 nM. FFA2 agonist-1 exhibits activity in β-arrestin-2 recruitment assay and cAMP inhibition assay with EC50 of 1.2 μM and 0.53 μM. FFA2 agonist-1 leads to appetite regulating peptide YY (PYY) mucosal responses, inhibits the fat accumulation, intestinal functions and food intake, and can be used for obesity research. | |||||||||||||||||||||
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