1394121-05-1
1394121-05-1
Chemical Structure
GNE 2861
- CAS No.: 1394121-05-1
- Formula:C22H26N6O2
- Molecular Weight:406.48
IUPAC Name: 1-((1-(2-aminopyrimidin-4-yl)-2-((2-methoxyethyl)amino)-1H-benzo[d]imidazol-6-yl)ethynyl)cyclohexan-1-ol
InChIKey: RZXMIHOUHYSGJO-UHFFFAOYSA-N
SMILES: OC1(C#CC2=CC=C3N=C(NCCOC)N(C4=NC(N)=NC=C4)C3=C2)CCCCC1
Biological Activity: GNE 2861 is a PAK inhibitor that displays group II selectivity. GNE 2861 inhibits PAK4, PAK5 and PAK6 with IC50s of 7.5, 36, 126 nM, respectively.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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GNE 2861 | 98.97% | GNE 2861 is a PAK inhibitor that displays group II selectivity. GNE 2861 inhibits PAK4, PAK5 and PAK6 with IC50s of 7.5, 36, 126 nM, respectively. | ||||||||||||||||||||
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