144980-77-8
Chemical Structure
Repinotan hydrochloride
Synonym(s): BAY x 3702
- CAS No.: 144980-77-8
- Formula:C21H25ClN2O4S
- Molecular Weight:436.95
IUPAC Name: (R)-2-(4-((chroman-2-ylmethyl)amino)butyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide hydrochloride
InChIKey: IGKYREHZJIHPML-UNTBIKODSA-N
SMILES: O=C(C1=C2C=CC=C1)N(CCCCNC[C@H]3CCC4=CC=CC=C4O3)S2(=O)=O.[H]Cl
Biological Activity: Repinotan hydrochloride (BAY x 3702) is a potent, selective, brain-penetrant and orally active 5-HT1A receptor agonist, with Ki values of 0.19 nM (calf hippocampus), 0.25 nM (rat and human cortex), and 0.59 nM (rat hippocampus Repinotan hydrochloride has a weak affinity for other related receptors. Repinotan hydrochloride has pronounced neuroprotective effects[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Repinotan hydrochloride | 97.08% | Repinotan hydrochloride (BAY x 3702) is a potent, selective, brain-penetrant and orally active 5-HT1A receptor agonist, with Ki values of 0.19 nM (calf hippocampus), 0.25 nM (rat and human cortex), and 0.59 nM (rat hippocampus Repinotan hydrochloride has a weak affinity for other related receptors. Repinotan hydrochloride has pronounced neuroprotective effects. | ||||||||||||||||||||
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