1451993-15-9
1451993-15-9
Chemical Structure
VU0467154
- CAS No.: 1451993-15-9
- Formula:C17H15F3N4O3S2
- Molecular Weight:444.45
IUPAC Name: 5-amino-3,4-dimethyl-N-(4-((trifluoromethyl)sulfonyl)benzyl)thieno[2,3-c]pyridazine-6-carboxamide
InChIKey: UDSFKIFLJPECRN-UHFFFAOYSA-N
SMILES: O=C(C1=C(N)C2=C(C)C(C)=NN=C2S1)NCC3=CC=C(S(=O)(C(F)(F)F)=O)C=C3
Biological Activity: VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor (mAChR), potentiating the response to ACh with pEC50s of 7.75, 6.2 and 6 for rat, human and cynomolgus monkey M4 receptor, respectively.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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VU0467154 | 99.23% | VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor (mAChR), potentiating the response to ACh with pEC50s of 7.75, 6.2 and 6 for rat, human and cynomolgus monkey M4 receptor, respectively. | ||||||||||||||||||||
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