1503332-97-5
1503332-97-5
Chemical Structure
EPZ020809
- CAS No.: 1503332-97-5
- Formula:C10H8N2O2
- Molecular Weight:188.18
InChIKey: RKSPSQDURYMIDD-UHFFFAOYSA-N
SMILES: O=C(C1=CC=NC(C2=CC=CN2)=C1)O
Biological Activity: EPZ020809 is a competitive KDM4C inhibitor with a Ki of 31 nM[1][2][3].
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EPZ020809 | EPZ020809 is a competitive KDM4C inhibitor with a Ki of 31 nM. | |||||||||||||||||||||
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References
- [1]. Das ND, et al. Chemical Inhibitors Targeting the Histone Lysine Demethylase Families with Potential for Drug Discovery. Epigenomes. 2023;7(1):7. Published 2023 Mar 11. [Content Brief]
- [2]. Wu Q, et al. Recent Advances with KDM4 Inhibitors and Potential Applications. J Med Chem. 2022;65(14):9564-9579. [Content Brief]
- [3]. Wigle TJ, et al. A High-Throughput Mass Spectrometry Assay Coupled with Redox Activity Testing Reduces Artifacts and False Positives in Lysine Demethylase Screening. J Biomol Screen. 2015;20(6):810-820. [Content Brief]
