153436-38-5
153436-38-5
Chemical Structure
Gavestinel sodium salt
Synonym(s): GV 150526A
- CAS No.: 153436-38-5
- Formula:C18H11Cl2N2NaO3
- Molecular Weight:397.19
IUPAC Name: sodium (E)-4,6-dichloro-3-(3-oxo-3-(phenylamino)prop-1-en-1-yl)-1H-indole-2-carboxylate
InChIKey: GRSDSTMFQHAESM-UHDJGPCESA-M
SMILES: O=C(NC1=CC=CC=C1)/C=C/C2=C(C(O[Na])=O)NC3=CC(Cl)=CC(Cl)=C23
Biological Activity: Gavestinel (GV 150526A) is a potent, selective, orally active and non-competitive antagonist of NMDA receptor. Gavestinel binds to the glycine site of the NMDA receptor, with a pKi of 8.5. Gavestinel can be used for the research of acute ischemic stroke[1].
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Gavestinel sodium salt | 98.58% | Gavestinel (GV 150526A) is a potent, selective, orally active and non-competitive antagonist of NMDA receptor. Gavestinel binds to the glycine site of the NMDA receptor, with a pKi of 8.5. Gavestinel can be used for the research of acute ischemic stroke. | ||||||||||||||||||||
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