158942-04-2
Chemical Structure
SB 206553
- CAS No.: 158942-04-2
- Formula:C17H16N4O
- Molecular Weight:292.34
IUPAC Name: 5-methyl-N-(pyridin-3-yl)-3,5-dihydropyrrolo[2,3-f]indole-1(2H)-carboxamide
InChIKey: QJQORSLQNXDVGE-UHFFFAOYSA-N
SMILES: O=C(N1CCC2=C1C=C3C(N(C)C=C3)=C2)NC4=CC=CN=C4
Biological Activity: SB 206553 is a 5-HT2C inverse agonist. SB 206553 can attenuate methamphetamine-seeking in rats. SB 206553 has activity for 5-HT2 receptor ligands in HEK-293 or CHO-K1 cells expressing human recombinant 5-HT2 receptors with pKi values of 5.6 nM (5-HT2A), 7.7 nM (5-HT2B) and 7.8 nM (5-HT2C), respectively. SB 206553 can be used for the research of psychostimulant abuse disorders[1].
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SB 206553 | 99.35% | SB 206553 is a 5-HT2C inverse agonist. SB 206553 can attenuate methamphetamine-seeking in rats. SB 206553 has activity for 5-HT2 receptor ligands in HEK-293 or CHO-K1 cells expressing human recombinant 5-HT2 receptors with pKi values of 5.6 nM (5-HT2A), 7.7 nM (5-HT2B) and 7.8 nM (5-HT2C), respectively. SB 206553 can be used for the research of psychostimulant abuse disorders. | ||||||||||||||||||||
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