1610362-93-0
Chemical Structure
APA-H-MPO hydrochloride
- CAS No.: 1610362-93-0
- Formula:C9H16ClN3O2
- Molecular Weight:233.70
IUPAC Name: 2-((3-aminopropyl)amino)-5-(hydroxymethyl)pyridine 1-oxide hydrochloride
InChIKey: UVXQESDWLUBIII-UHFFFAOYSA-N
SMILES: OCC1=CC=C([N+]([O-])=C1)NCCCN.[H]Cl
Biological Activity: APA-H-MPO hydrochloride is an inhibitor of PCAF bromodomain/Tat-AcK50 interaction with potential for anti-HIV/AIDS. APA-H-MPO hydrochloride can effectively inhibit the binding of PCAF bromodomain to Tat-AcK50. APA-H-MPO hydrochloride showed low cytotoxicity in preliminary cell studies. APA-H-MPO hydrochloride is considered a potential candidate for a promising inhibitory strategy targeting the host cell protein PCAF BRD to block HIV replication[1].
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APA-H-MPO hydrochloride | APA-H-MPO hydrochloride is an inhibitor of PCAF bromodomain/Tat-AcK50 interaction with potential for anti-HIV/AIDS. APA-H-MPO hydrochloride can effectively inhibit the binding of PCAF bromodomain to Tat-AcK50. APA-H-MPO hydrochloride showed low cytotoxicity in preliminary cell studies. APA-H-MPO hydrochloride is considered a potential candidate for a promising inhibitory strategy targeting the host cell protein PCAF BRD to block HIV replication. | |||||||||||||||||||||
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