1643879-88-2
1643879-88-2
Chemical Structure
NTRC-808
- CAS No.: 1643879-88-2
- Formula:C23H24ClN3O5
- Molecular Weight:457.91
IUPAC Name: (6-chloro-4-(2,6-dimethoxyphenyl)quinazoline-2-carbonyl)-L-leucine
InChIKey: QRMVAUUKTYTTEN-INIZCTEOSA-N
SMILES: CC(C)C[C@@H](C(O)=O)NC(C1=NC(C2=C(OC)C=CC=C2OC)=C3C=C(Cl)C=CC3=N1)=O
Biological Activity: NTRC-808 is a nonpeptide selective GPCR neurotensin receptor type 2 (NTS2) partial agonist with an EC50 of 14 nM and Ki of 88 nM. NTRC-808 has higher selectivity for NTS2 than for NTS1. NTRC-808 has antipsychotic and analgesic activity[1].
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NTRC-808 | NTRC-808 is a nonpeptide selective GPCR neurotensin receptor type 2 (NTS2) partial agonist with an EC50 of 14 nM and Ki of 88 nM. NTRC-808 has higher selectivity for NTS2 than for NTS1. NTRC-808 has antipsychotic and analgesic activity. | |||||||||||||||||||||
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