171549-56-7
171549-56-7
Chemical Structure
GR-4991W93
- CAS No.: 171549-56-7
- Formula:C18H23N3O2
- Molecular Weight:313.39
IUPAC Name: (S)-4-((3-((1r,3S)-3-(dimethylamino)cyclobutyl)-1H-indol-5-yl)methyl)oxazolidin-2-one
InChIKey: JLDUTSKKXXJGGG-IHRRRGAJSA-N
SMILES: CN(C)[C@H](C1)C[C@@H]1C2=CNC3=CC=C(C[C@@H]4NC(OC4)=O)C=C32
Biological Activity: GR-4991W93 is an orally active partial agonist against 5HT1B/1D receptor, with pIC50 values of 6.95 and 7.80 against 5HT1B and 5HT1D, respectively. GR-4991W93 demonstrates potent inhibition of electrically evoked plasma extravasation in the guinea pig. GR-4991W93 can be used for migraine research[1].
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GR-4991W93 | GR-4991W93 is an orally active partial agonist against 5HT1B/1D receptor, with pIC50 values of 6.95 and 7.80 against 5HT1B and 5HT1D, respectively. GR-4991W93 demonstrates potent inhibition of electrically evoked plasma extravasation in the guinea pig. GR-4991W93 can be used for migraine research. | |||||||||||||||||||||
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