182633-59-6
182633-59-6
Chemical Structure
LY320954
- CAS No.: 182633-59-6
- Formula:C21H26N4O3
- Molecular Weight:382.46
IUPAC Name: (E)-2-(4-((3-hydroxy-4-propionyl-2-propylbenzyl)oxy)benzylidene)hydrazine-1-carboximidamide
InChIKey: TUJFUBGJRSXFHG-WYMPLXKRSA-N
SMILES: CCCC1=C(O)C(C(CC)=O)=CC=C1COC2=CC=C(/C=N/NC(N)=N)C=C2
Biological Activity: LY320954 is a selective 5-HT2A receptor antagonist, with a Ki of 96 nM. LY320954 potently inhibits Ca2+ influx in the functional assay (EC50 of 35.5 nM). LY320954 inhibits 5-HT-induced paw swelling in rats, with ED50 of 4.8 mg/kg[1].
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LY320954 | LY320954 is a selective 5-HT2A receptor antagonist, with a Ki of 96 nM. LY320954 potently inhibits Ca2+ influx in the functional assay (EC50 of 35.5 nM). LY320954 inhibits 5-HT-induced paw swelling in rats, with ED50 of 4.8 mg/kg. | |||||||||||||||||||||
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