1854061-19-0
1854061-19-0
Chemical Structure
PF-06761281
- CAS No.: 1854061-19-0
- Formula:C13H17NO6
- Molecular Weight:283.28
IUPAC Name: (R)-2-hydroxy-2-(2-(2-methoxy-5-methylpyridin-3-yl)ethyl)succinic acid
InChIKey: FGYMJXFSHBLHLW-CYBMUJFWSA-N
SMILES: O=C(O)[C@](CCC1=CC(C)=CN=C1OC)(O)CC(O)=O
Biological Activity: PF-06761281 (Compound 4a) is a potent, orally active, partial selective sodium-coupled citrate transporter (NaCT or SLC13A5) inhibitor with IC50 values of 0.51, 13.2 and 14.1 µM against HEKNaCT, HEKNaDC1 and HEKNaDC3, respectively[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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PF-06761281 | 99.52% | PF-06761281 (Compound 4a) is a potent, orally active, partial selective sodium-coupled citrate transporter (NaCT or SLC13A5) inhibitor with IC50 values of 0.51, 13.2 and 14.1 µM against HEKNaCT, HEKNaDC1 and HEKNaDC3, respectively. | ||||||||||||||||||||
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