1934301-68-4
1934301-68-4
Chemical Structure
MRK-A
- CAS No.: 1934301-68-4
- Formula:C28H30N4O2
- Molecular Weight:454.56
IUPAC Name: (8-morpholino-5,11-dihydro-6H-benzo[b]pyrido[2,3-e][1,4]diazepin-6-yl)(6,7,8,9-tetrahydro-5H-benzo[7]annulen-7-yl)methanone
InChIKey: ZGJIUUQQZUDAKL-UHFFFAOYSA-N
SMILES: O=C(N1CC2=CC=CN=C2NC3=CC=C(N4CCOCC4)C=C13)C5CCC6=CC=CC=C6CC5
Biological Activity: MRK-A is a selective, blood-brain-barrier permeable mutant IDH1 inhibitor with an IC50 value of 5 nM. MRK-A inhibits 2-HG production. MRK-A has anti-cancer activity against brain tumors[1].
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MRK-A | MRK-A is a selective, blood-brain-barrier permeable mutant IDH1 inhibitor with an IC50 value of 5 nM. MRK-A inhibits 2-HG production. MRK-A has anti-cancer activity against brain tumors. | |||||||||||||||||||||
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