1952261-87-8
1952261-87-8
Chemical Structure
EP3 antagonist 2
- CAS No.: 1952261-87-8
- Formula:C21H21N3O2
- Molecular Weight:347.41
IUPAC Name: (R)-3-(3-methyl-2-oxopiperidin-3-yl)-6-(5-methylquinolin-3-yl)pyridin-2(1H)-one
InChIKey: OJVNYQOKTZLPPX-OAQYLSRUSA-N
SMILES: O=C1C([C@]2(C)C(NCCC2)=O)=CC=C(C3=CC4=C(C)C=CC=C4N=C3)N1
Biological Activity: EP3 antagonist 2 (Compound Exp 1) is a potent and selective EP3 receptor antagonist. EP3 antagonist 2 has a strong binding affinity for the human EP3 receptor (Ki: 3.3 nM) and significant antagonistic activity (IC50: 30.8 nM, determined by cellular cAMP levels)[1].
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EP3 antagonist 2 | EP3 antagonist 2 (Compound Exp 1) is a potent and selective EP3 receptor antagonist. EP3 antagonist 2 has a strong binding affinity for the human EP3 receptor (Ki: 3.3 nM) and significant antagonistic activity (IC50: 30.8 nM, determined by cellular cAMP levels). | |||||||||||||||||||||
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