2055015-61-5
2055015-61-5
Chemical Structure
GLPG2451
- CAS No.: 2055015-61-5
- Formula:C16H16F3N3O5S
- Molecular Weight:419.38
IUPAC Name: (S)-3-amino-N-(2-hydroxypropyl)-5-((4-(trifluoromethoxy)phenyl)sulfonyl)picolinamide
InChIKey: UMOGNCVNHXWFIX-VIFPVBQESA-N
SMILES: O=S(C1=CC=C(OC(F)(F)F)C=C1)(C2=CN=C(C(NC[C@@H](O)C)=O)C(N)=C2)=O
Biological Activity: GLPG2451 is a cystic fibrosis transmembrane conductance regulator (CFTR) potentiator, which effectively potentiates low temperature rescued F508del CFTR with an EC50 of 11.1 nM[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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GLPG2451 | 99.25% | GLPG2451 is a cystic fibrosis transmembrane conductance regulator (CFTR) potentiator, which effectively potentiates low temperature rescued F508del CFTR with an EC50 of 11.1 nM. | ||||||||||||||||||||
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