2079896-25-4
2079896-25-4
Chemical Structure
GSK 4027
- CAS No.: 2079896-25-4
- Formula:C17H21BrN4O
- Molecular Weight:377.28
IUPAC Name: 4-bromo-2-methyl-5-(((3R,5R)-1-methyl-5-phenylpiperidin-3-yl)amino)pyridazin-3(2H)-one
InChIKey: VZAFGXCWAWRULT-UONOGXRCSA-N
SMILES: BrC1=C(N[C@@H]2C[C@H](C3=CC=CC=C3)CN(C)C2)C=NN(C)C1=O
Biological Activity: GSK 4027 is a chemical probe for the PCAF/GCN5 bromodomain with an pIC50 of 7.4±0.11 for PCAF in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay.
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GSK 4027 | 98.22% | GSK 4027 is a chemical probe for the PCAF/GCN5 bromodomain with an pIC50 of 7.4±0.11 for PCAF in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. | ||||||||||||||||||||
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GSK 4027 (Standard) | ≥98% | GSK 4027 (Standard) is the analytical standard of GSK 4027 (HY-101027). This product is intended for research and analytical applications. GSK 4027 is a chemical probe for the PCAF/GCN5 bromodomain with an pIC50 of 7.4±0.11 for PCAF in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. | ||||||||||||||||||||
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