2093408-03-6
2093408-03-6
Chemical Structure
AY254
- CAS No.: 2093408-03-6
- Formula:C30H49N9O6
- Molecular Weight:631.77
InChIKey: ZVDSAIOSGOWYAW-CKLTXHEASA-N
SMILES: O=C(C1=CC=NO1)N[C@@H](CC2CCCCC2)C(N[C@@H](C3CCCCC3)C(N[C@@H](C)C(N[C@H](C(N)=O)CCCNC(N)=N)=O)=O)=O
Biological Activity: AY254 is an analogue of AY77 (HY-138951). AY254 is ERK-biased PAR2 agonist with an EC50 of 2 nM. AY254 relieves cytokine-induced caspase 3/8 activation. AY254 also promotes scratch-wound healing and induced IL-8 secretion via PAR2-ERK1/2 signaling[1]
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AY254 | AY254 is an analogue of AY77 (HY-138951). AY254 is ERK-biased PAR2 agonist with an EC50 of 2 nM. AY254 relieves cytokine-induced caspase 3/8 activation. AY254 also promotes scratch-wound healing and induced IL-8 secretion via PAR2-ERK1/2 signaling | |||||||||||||||||||||
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