2158201-04-6
2158201-04-6
Chemical Structure
Cav 3.1 blocker 1
- CAS No.: 2158201-04-6
- Formula:C26H19F6N3O2
- Molecular Weight:519.44
InChIKey: RJAGHFCAXLPKOE-UHFFFAOYSA-N
SMILES: O=C(C1=NN(C(C2=CC=CC=C2)=C1C(F)F)C3=CC=C(C=C3)F)NCC4=C(OCC(F)(F)F)C=CC=C4
Biological Activity: Cav 3.1 blocker 1 (compound 12) is a T-type calcium channel blocker with an IC50value of 160 nM for Cav3.1. Cav 3.1 blocker 1 weakly inhibits Cav 3.2 (IC50 of 5000 nM), and shows no inhibition on Cav 3.3 and Cav 1.2 (IC50 of >10000 nM)[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Cav 3.1 blocker 1 | Cav 3.1 blocker 1 (compound 12) is a T-type calcium channel blocker with an IC50value of 160 nM for Cav3.1. Cav 3.1 blocker 1 weakly inhibits Cav 3.2 (IC50 of 5000 nM), and shows no inhibition on Cav 3.3 and Cav 1.2 (IC50 of >10000 nM). | |||||||||||||||||||||
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