2309762-29-4
2309762-29-4
Chemical Structure
Elacestrant (S enantiomer)
Synonym(s): RAD1901 S enantiomer
- CAS No.: 2309762-29-4
- Formula:C30H38N2O2
- Molecular Weight:458.63
IUPAC Name: (S)-6-(2-(ethyl(4-(2-(ethylamino)ethyl)benzyl)amino)-4-methoxyphenyl)-5,6,7,8-tetrahydronaphthalen-2-ol
InChIKey: SIFNOOUKXBRGGB-SANMLTNESA-N
SMILES: OC1=CC=C2C[C@@H](C3=CC=C(OC)C=C3N(CC)CC4=CC=C(CCNCC)C=C4)CCC2=C1
Biological Activity: Elacestrant S enantiomer (RAD1901 S enantiomer) is an low activity enantiomer of elacestrant. Elacestrant (RAD1901) is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Elacestrant (S enantiomer) | 94.65% | Elacestrant S enantiomer (RAD1901 S enantiomer) is an low activity enantiomer of elacestrant. Elacestrant (RAD1901) is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively. | ||||||||||||||||||||
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