2316832-86-5
2316832-86-5
Chemical Structure
ERRγ inverse agonist 1
- CAS No.: 2316832-86-5
- Formula:C30H38Cl2N2O2
- Molecular Weight:529.54
IUPAC Name: (E)-3-(5-hydroxy-1-(4-(4-isopropylpiperazin-1-yl)phenyl)-2-phenylpent-1-en-1-yl)phenol dihydrochloride
InChIKey: VREKGOHYUPVQSX-NFOZGECASA-N
SMILES: OC1=CC=CC(/C(C2=CC=C(N3CCN(C(C)C)CC3)C=C2)=C(C4=CC=CC=C4)\CCCO)=C1.[H]Cl.[H]Cl
Biological Activity: ERRγ inverse agonist 1 (Compound 12) is a selective ERRγ inverse agonist with an IC50 value of 0.040 μM against ERRγ. ERRγ inverse agonist 1 inhibits the activity of ERRγ at the functional level. ERRγ inverse agonist 1 can be used in the research of anaplastic thyroid cancer[1].
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ERRγ inverse agonist 1 | ERRγ inverse agonist 1 (Compound 12) is a selective ERRγ inverse agonist with an IC50 value of 0.040 μM against ERRγ. ERRγ inverse agonist 1 inhibits the activity of ERRγ at the functional level. ERRγ inverse agonist 1 can be used in the research of anaplastic thyroid cancer. | |||||||||||||||||||||
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