2395016-49-4
2395016-49-4
Chemical Structure
P2Y2R/GPR17 antagonist 1
- CAS No.: 2395016-49-4
- Formula:C19H13ClN2O6S
- Molecular Weight:432.83
IUPAC Name: 3-nitrophenyl 4-(2-chlorobenzamido)benzenesulfonate
InChIKey: YGSIMJKEUKTDFX-UHFFFAOYSA-N
SMILES: O=C(C1=C(C=CC=C1)Cl)NC2=CC=C(C=C2)S(=O)(OC3=CC([N+]([O-])=O)=CC=C3)=O
Biological Activity: P2Y2R/GPR17 antagonist 1 (Compound 14m) is a dual P2Y2R and GPR17 antagonist with IC50 values of 3.17 µM and 1.67 µM against P2Y2R and GPR17, respectively. P2Y2R/GPR17 antagonist 1 shows excellent metabolic stability in human liver microsomes[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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P2Y2R/GPR17 antagonist 1 | 98.09% | P2Y2R/GPR17 antagonist 1 (Compound 14m) is a dual P2Y2R and GPR17 antagonist with IC50 values of 3.17 µM and 1.67 µM against P2Y2R and GPR17, respectively. P2Y2R/GPR17 antagonist 1 shows excellent metabolic stability in human liver microsomes. | ||||||||||||||||||||
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