2410557-00-3
2410557-00-3
Chemical Structure
iRucaparib-AP6
- CAS No.: 2410557-00-3
- Formula:C46H55FN6O11
- Molecular Weight:886.96
IUPAC Name: 2-(2,6-dioxopiperidin-3-yl)-4-((1-(4-(8-fluoro-1-oxo-2,3,4,6-tetrahydro-1H-azepino[5,4,3-cd]indol-5-yl)phenyl)-2-methyl-5,8,11,14,17,20-hexaoxa-2-azadocosan-22-yl)amino)isoindoline-1,3-dione
InChIKey: YHMDCINUVWULST-UHFFFAOYSA-N
SMILES: O=C(NCC1)C2=CC(F)=CC3=C2C1=C(C4=CC=C(C=C4)CN(CCOCCOCCOCCOCCOCCOCCNC5=CC=CC(C(N6C7CCC(NC7=O)=O)=O)=C5C6=O)C)N3
Biological Activity: iRucaparib-AP6 is a highly efficient and specific PROTAC PARP1 degrader. iRucaparib-AP6, a non-trapping PARP1 degrader, blocks both the catalytic activity and scaffolding effects of PARP1[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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iRucaparib-AP6 | 99.03% | iRucaparib-AP6 is a highly efficient and specific PROTAC PARP1 degrader. iRucaparib-AP6, a non-trapping PARP1 degrader, blocks both the catalytic activity and scaffolding effects of PARP1. | ||||||||||||||||||||
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