2410793-22-3

GRK5-IN-3 Chemical Structure
2410793-22-3

Chemical Structure

GRK5-IN-3

  • CAS No.: 2410793-22-3
  • Formula:C23H21N7O3
  • Molecular Weight:443.46

IUPAC Name: 2-((2-((4-acrylamido-2-methoxyphenyl)amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino)benzamide

InChIKey: PYFNYNPQSUXBGV-UHFFFAOYSA-N

SMILES: O=C(NC1=CC=C(C(OC)=C1)NC2=NC(NC3=C(C(N)=O)C=CC=C3)=C4C=CNC4=N2)C=C

Biological Activity: GRK5-IN-3 is a covalent inhibitor of GRK5 (G Protein-Coupled Receptor Kinase 5). GRK5-IN-3 shows potent inhibitory effect to GRK5 and GRK6 with IC50s of 0.22 μM and 0.41 μM, respectively[1].

Cat. No. Product Name Purity Description Pricing
HY-150021
GRK5-IN-3 GRK5-IN-3 is a covalent inhibitor of GRK5 (G Protein-Coupled Receptor Kinase 5). GRK5-IN-3 shows potent inhibitory effect to GRK5 and GRK6 with IC50s of 0.22 μM and 0.41 μM, respectively.
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This product is a controlled substance and not for sale in your territory.

This product is not for sale in your territory.

This compound is listed in the SVHC (Substances of Very High Concern) candidate list of ECHA (European Chemicals Agency).

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References