2411088-16-7
2411088-16-7
Chemical Structure
5-HT6/5-HT2A receptor ligand-2
- CAS No.: 2411088-16-7
- Formula:C20H18FN3O2
- Molecular Weight:351.37
IUPAC Name: 4-(5-(((2-(5-fluoro-1H-pyrrolo[2,3-b]pyridin-3-yl)ethyl)amino)methyl)furan-2-yl)phenol
InChIKey: VTRMFVAGEAFJTR-UHFFFAOYSA-N
SMILES: OC1=CC=C(C2=CC=C(CNCCC3=CNC4=NC=C(F)C=C43)O2)C=C1
Biological Activity: 5-HT6/5-HT2A receptor ligand-2 (compound 42) is a brain-penetrant dual 5-HT6/5-HT2A receptor antagonist, with a Ki of 25 nM and 32 nM, respectively. 5-HT6/5-HT2A receptor ligand-2 shows pro-cognitive properties[1].
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5-HT6/5-HT2A receptor ligand-2 | 5-HT6/5-HT2A receptor ligand-2 (compound 42) is a brain-penetrant dual 5-HT6/5-HT2A receptor antagonist, with a Ki of 25 nM and 32 nM, respectively. 5-HT6/5-HT2A receptor ligand-2 shows pro-cognitive properties. | |||||||||||||||||||||
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