2420551-38-6
2420551-38-6
Chemical Structure
ERAP2-IN-1
- CAS No.: 2420551-38-6
- Formula:C20H21F3N2O5S
- Molecular Weight:458.45
IUPAC Name: 4-methoxy-3-(N-(2-(piperidin-1-yl)-4-(trifluoromethyl)phenyl)sulfamoyl)benzoic acid
InChIKey: BGLAMEXMBJAJBI-UHFFFAOYSA-N
SMILES: O=C(O)C1=CC=C(OC)C(S(=O)(NC2=CC=C(C(F)(F)F)C=C2N3CCCCC3)=O)=C1
Biological Activity: ERAP2-IN-1 (compound 61) is an uncompetitive ERAP2 inhibitor. ERAP2-IN-1 specifically inhibits the ERAP2 peptide hydrolysis activity, inhibiting Arg-AMC hydrolysis with an IC50 of 27 μM and model peptide hydrolysis with an IC50 of 44 μM[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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ERAP2-IN-1 | 98.86% | ERAP2-IN-1 (compound 61) is an uncompetitive ERAP2 inhibitor. ERAP2-IN-1 specifically inhibits the ERAP2 peptide hydrolysis activity, inhibiting Arg-AMC hydrolysis with an IC50 of 27 μM and model peptide hydrolysis with an IC50 of 44 μM. | ||||||||||||||||||||
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