2447039-81-6
Chemical Structure
RAS/RAS-RAF-IN-1
- CAS No.: 2447039-81-6
- Formula:C45H57N7O7
- Molecular Weight:807.98
IUPAC Name: (3S)-1-acryloyl-N-((2S)-1-(((63S,4S)-13-(2-cyanopropan-2-yl)-25-hydroxy-10,10-dimethyl-5,7-dioxo-61,62,63,64,65,66-hexahydro-11H-8-oxa-1(6,1)-indola-6(1,3)-pyridazina-2(1,3)-benzenacycloundecaphane-4-yl)amino)-3-methyl-1-oxobutan-2-yl)-N-methylpyrrolidine
InChIKey: RCXSKUOUWMZVFF-NXCZKTMTSA-N
SMILES: CC(C)(C1=CN(CC(C)(COC([C@@](CCC2)([H])NN2C3=O)=O)C)C4=CC(C5=CC(O)=CC(C[C@@H]3NC([C@H](C(C)C)N(C)C([C@@H](CC6)CN6C(C=C)=O)=O)=O)=C5)=CC=C41)C#N
Biological Activity: RAS/RAS-RAF-IN-1 is a potent RAS and RAS-RAF inhibitor. RAS/RAS-RAF-IN-1 has a KD of 5.0 μΜ-15 μΜ for cyclophilin A (CYPA) binding affinity. RAS/RAS-RAF-IN-1 has antitumor activity[1].
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RAS/RAS-RAF-IN-1 | RAS/RAS-RAF-IN-1 is a potent RAS and RAS-RAF inhibitor. RAS/RAS-RAF-IN-1 has a KD of 5.0 μΜ-15 μΜ for cyclophilin A (CYPA) binding affinity. RAS/RAS-RAF-IN-1 has antitumor activity. | |||||||||||||||||||||
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