2490311-14-1
Chemical Structure
BRD4 Inhibitor-20
- CAS No.: 2490311-14-1
- Formula:C18H18N2O4S
- Molecular Weight:358.41
IUPAC Name: 2-methoxy-N-(2-oxo-3-(propan-2-ylidene)indolin-5-yl)benzenesulfonamide
InChIKey: CDERLIUJSXSXFH-UHFFFAOYSA-N
SMILES: O=C1NC2=CC=C(C=C2/C1=C(C)\C)NS(=O)(C3=C(C=CC=C3)OC)=O
Biological Activity: BRD4 Inhibitor-20 is a potent orally active bromodomain protein 4 (BRD4) inhibitor. BRD4 Inhibitor-20 has inhibitory activity for BRD4 (BD1) and BRD4 (BD2) with IC50 values of 19 nM and 28 nM, respectively. BRD4 Inhibitor-20 also has anti-proliferation activities in cancer cell lines. BRD4 Inhibitor-20 can be used for the research of kinds of cancer, such as colon cancer[1].
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BRD4 Inhibitor-20 | 99.24% | BRD4 Inhibitor-20 is a potent orally active bromodomain protein 4 (BRD4) inhibitor. BRD4 Inhibitor-20 has inhibitory activity for BRD4 (BD1) and BRD4 (BD2) with IC50 values of 19 nM and 28 nM, respectively. BRD4 Inhibitor-20 also has anti-proliferation activities in cancer cell lines. BRD4 Inhibitor-20 can be used for the research of kinds of cancer, such as colon cancer. | ||||||||||||||||||||
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