2638507-71-6
2638507-71-6
Chemical Structure
EP300/CBP-IN-1
- CAS No.: 2638507-71-6
- Formula:C30H32ClFN4O4
- Molecular Weight:567.05
InChIKey: SOVZFVKUVPGESE-CLHVYKLBSA-N
SMILES: O=C1N(C2=CC(F)=C(C=C2)Cl)[C@@H](CCO1)C3=NC4=CC(C5=C(C)ON=C5C)=CC=C4N3[C@H]6CC[C@@H](CC6)OCC
Biological Activity: EP300/CBP-IN-1 (compound 172) is a potent EP300/CBP inhibitor with IC50s of 2.3 nM and 2.1 nM for CBP BRD and EP300 BRD, respectively. EP300/CBP-IN-1 has the inhibitory effect on the proliferation of prostate cancer CWR22RV1 cells[1].
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EP300/CBP-IN-1 | EP300/CBP-IN-1 (compound 172) is a potent EP300/CBP inhibitor with IC50s of 2.3 nM and 2.1 nM for CBP BRD and EP300 BRD, respectively. EP300/CBP-IN-1 has the inhibitory effect on the proliferation of prostate cancer CWR22RV1 cells. | |||||||||||||||||||||
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