2654075-81-5
2654075-81-5
Chemical Structure
H-APPAMP-003
- CAS No.: 2654075-81-5
- Formula:C23H30N8O
- Molecular Weight:434.54
InChIKey: JWLYZTFPPDFIIV-APWZRJJASA-N
SMILES: CC(C1=C2N=C(NC[C@H]3CCNC[C@@H]3O)C=C(NCC4=CN5C=CC=CC5=N4)N2N=C1)C
Biological Activity: H-APPAMP-003 is a CDK12 inhibitor with an IC50 of 50.2 nM. H-APPAMP-003 shows weak inhibition of CDK7 with an IC50 of 411 nM. H-APPAMP-003 is also a molecular glue[1].
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H-APPAMP-003 | H-APPAMP-003 is a CDK12 inhibitor with an IC50 of 50.2 nM. H-APPAMP-003 shows weak inhibition of CDK7 with an IC50 of 411 nM. H-APPAMP-003 is also a molecular glue. | |||||||||||||||||||||
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