2752378-78-0
2752378-78-0
Chemical Structure
RXFP3/4 agonist 2
- CAS No.: 2752378-78-0
- Formula:C22H22N6O2
- Molecular Weight:402.45
IUPAC Name: methyl (E)-4-(2-(2-((5-cyano-7-methyl-1H-indol-3-yl)methylene)hydrazine-1-carboximidamido)ethyl)benzoate
InChIKey: XIVYUSRYHWXGLX-UVHMKAGCSA-N
SMILES: COC(C(C=C1)=CC=C1CCNC(N/N=C/C(C2=CC(C#N)=C3)=CNC2=C3C)=N)=O
Biological Activity: RXFP3/4 agonist 2 is a potent, nonpeptide dual RXFP3/4 agonist (EC50=3.1 and 2.7 nM). RXFP3/4 agonist 2 also potently promotes interactions between RXFP3 and β-arrestin-2 with EC50 values in the range of 10-22 nM[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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RXFP3/4 agonist 2 | 99.75% | RXFP3/4 agonist 2 is a potent, nonpeptide dual RXFP3/4 agonist (EC50=3.1 and 2.7 nM). RXFP3/4 agonist 2 also potently promotes interactions between RXFP3 and β-arrestin-2 with EC50 values in the range of 10-22 nM. | ||||||||||||||||||||
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