2760307-53-5
2760307-53-5
Chemical Structure
BRD4 Inhibitor-23
- CAS No.: 2760307-53-5
- Formula:C22H19F2N3O4S
- Molecular Weight:459.47
IUPAC Name: 1-(2-(2,4-difluorophenoxy)-5-((ethylsulfonyl)methyl)pyridin-3-yl)-3-methyl-1,5-dihydro-4H-pyrrolo[3,2-c]pyridin-4-one
InChIKey: XJYPAGQKIHIXCO-UHFFFAOYSA-N
SMILES: CCS(=O)(CC1=CC(N2C=C(C3=C2C=CNC3=O)C)=C(N=C1)OC4=C(C=C(C=C4)F)F)=O
Biological Activity: BRD4 Inhibitor-23 is a potent and orally active BRD4 inhibitor with IC50s of 6.21 nM and 1.44 nM for BRD4 BD-1 and BRD4 BD-2, respectively (WO2022033542A1; Example 1)[1].
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BRD4 Inhibitor-23 | BRD4 Inhibitor-23 is a potent and orally active BRD4 inhibitor with IC50s of 6.21 nM and 1.44 nM for BRD4 BD-1 and BRD4 BD-2, respectively (WO2022033542A1; Example 1). | |||||||||||||||||||||
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