2819989-60-9
2819989-60-9
Chemical Structure
PBRM1-BD2-IN-4
- CAS No.: 2819989-60-9
- Formula:C15H13ClN2O
- Molecular Weight:272.73
InChIKey: ZDFFMEAQARQRHC-UHFFFAOYSA-N
SMILES: O=C1NC(C2=CC=CC=C2C)NC3=C1C(Cl)=CC=C3
Biological Activity: PBRM1-BD2-IN-4 is a PBRM1-BD2 inhibitor with an IC50 of 0.2 μM, and its Kd values for PBRM1-BD2 and PBRM1-BD5 are 5.5 μM and 11.1 μM, respectively. PBRM1-BD2-IN-4 selectively inhibits the proliferation of PBRM1-dependent prostate cancer cells. PBRM1-BD2-IN-4 can be used in studies related to prostate cancer[1].
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PBRM1-BD2-IN-4 | PBRM1-BD2-IN-4 is a PBRM1-BD2 inhibitor with an IC50 of 0.2 μM, and its Kd values for PBRM1-BD2 and PBRM1-BD5 are 5.5 μM and 11.1 μM, respectively. PBRM1-BD2-IN-4 selectively inhibits the proliferation of PBRM1-dependent prostate cancer cells. PBRM1-BD2-IN-4 can be used in studies related to prostate cancer. | |||||||||||||||||||||
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