2821085-76-9
2821085-76-9
Chemical Structure
CB2R/5-HT1AR agonist 1
- CAS No.: 2821085-76-9
- Formula:C24H33NO3
- Molecular Weight:383.52
InChIKey: LHZJDQKOCOLSNK-DLBZAZTESA-N
SMILES: CCCCC1(C2=C(C(O)=C([C@H]3[C@@H](CCC(C)=C3)C(C)=C)C(O)=C2)C(N)=O)CC1
Biological Activity: CB2R/5-HT1AR agonist 1 (Compound 2o) is an orally active partial agonist of the CB2 receptor (EC50=479.6 nM). CB2R/5-HT1AR agonist 1 is a full agonist of 5-HT1A receptor (EC50=2.7 μM). CB2R/5-HT1AR agonist 1 exhibits anti-anxiety and anti-depressive effects. CB2R/5-HT1AR agonist 1 possesses favorable pharmacokinetic properties[1].
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CB2R/5-HT1AR agonist 1 | CB2R/5-HT1AR agonist 1 (Compound 2o) is an orally active partial agonist of the CB2 receptor (EC50=479.6 nM). CB2R/5-HT1AR agonist 1 is a full agonist of 5-HT1A receptor (EC50=2.7 μM). CB2R/5-HT1AR agonist 1 exhibits anti-anxiety and anti-depressive effects. CB2R/5-HT1AR agonist 1 possesses favorable pharmacokinetic properties. | |||||||||||||||||||||
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