2833692-02-5
2833692-02-5
Chemical Structure
MOR agonist-2
- CAS No.: 2833692-02-5
- Formula:C37H47Cl2N5O3
- Molecular Weight:680.71
InChIKey: KZUQRBDBFQHGDF-NDKRRWIDSA-N
SMILES: O=C([C@H]1N(CCC(C2=CC=CC=C2)(C3=CC=CC=C3)C(N(C)C)=O)C[C@H](O)C1)NCCCCN4CCN(C5=CC=CC(Cl)=C5Cl)CC4
Biological Activity: MOR agonist-2 (compound 46) is a antagonist of D3R and agonist of MOR (Ki: 7.26 nM and 564 nM, respectively). MOR agonist-2 has the potential to produce analgesic effects through MOR partial agonism. MOR agonist-2 reduces opioid-misuse liability via D3R antagonism[1].
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MOR agonist-2 | MOR agonist-2 (compound 46) is a antagonist of D3R and agonist of MOR (Ki: 7.26 nM and 564 nM, respectively). MOR agonist-2 has the potential to produce analgesic effects through MOR partial agonism. MOR agonist-2 reduces opioid-misuse liability via D3R antagonism. | |||||||||||||||||||||
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