2839471-45-1
Chemical Structure
LPA5 antagonist 1
- CAS No.: 2839471-45-1
- Formula:C28H26N2O4S
- Molecular Weight:486.58
IUPAC Name: 4-(tert-butyl)-1,2,6,7-tetrahydro-8H-indeno[5,4-b]furan-8-one
InChIKey: KNTSYYKDKFNRKN-UHFFFAOYSA-N
SMILES: O=C1N(C2=CC=C3C(C(C)=CS3)=C2)C=C(C(N4CCC(C#C)CC4)=O)C5=C1C=C(OC)C(OC)=C5
Biological Activity: LPA5 antagonist 1 (Compound 66) is a potent and selective lysophosphatidic acid receptor 5 (LPA5) antagonist (IC50=32 nM). LPA5 antagonist 1 shows high blood-brain-barrier permeability and anti-nociceptive activity. LPA5 antagonist 1 can be used in inflammatory and neuropathic pain research[1]. LPA5 antagonist 1 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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LPA5 antagonist 1 | 98.91% | LPA5 antagonist 1 (Compound 66) is a potent and selective lysophosphatidic acid receptor 5 (LPA5) antagonist (IC50=32 nM). LPA5 antagonist 1 shows high blood-brain-barrier permeability and anti-nociceptive activity. LPA5 antagonist 1 can be used in inflammatory and neuropathic pain research. LPA5 antagonist 1 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups. | ||||||||||||||||||||
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