2848719-34-4
2848719-34-4
Chemical Structure
FAAH/MAGL-IN-3
- CAS No.: 2848719-34-4
- Formula:C21H25N3O6S
- Molecular Weight:447.50
IUPAC Name: 4-nitrophenyl 4-((4-butylphenyl)sulfonyl)piperazine-1-carboxylate
InChIKey: WSNBDRIOXKWWCY-UHFFFAOYSA-N
SMILES: CCCCC1=CC=C(C=C1)S(=O)(N2CCN(CC2)C(OC3=CC=C(C=C3)[N+]([O-])=O)=O)=O
Biological Activity: FAAH/MAGL-IN-3 (Compound 10) is an irreversible fatty acid amide hydrolase (FAAH) and monoacylglycerol lipase (MAGL) dual inhibitor with IC50 values of 179 and 759 nM against FAAH and MAGL, respectively. FAAH/MAGL-IN-3 shows low PAMPA (Parallel Artificial Membrane Permeability Assay) permeability[1].
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FAAH/MAGL-IN-3 | FAAH/MAGL-IN-3 (Compound 10) is an irreversible fatty acid amide hydrolase (FAAH) and monoacylglycerol lipase (MAGL) dual inhibitor with IC50 values of 179 and 759 nM against FAAH and MAGL, respectively. FAAH/MAGL-IN-3 shows low PAMPA (Parallel Artificial Membrane Permeability Assay) permeability. | |||||||||||||||||||||
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