2851993-77-4
2851993-77-4
Chemical Structure
RJG-2051
- CAS No.: 2851993-77-4
- Formula:C26H31N5O4S
- Molecular Weight:509.62
InChIKey: HMWIALSNZLCBBI-UHFFFAOYSA-N
SMILES: COC1=CC=CC=C1N2CCN(CC2)C(C3=CC=C(C=C3)S(=O)(N4C=NC(C5CCCCC5)=N4)=O)=O
Biological Activity: RJG-2051 is a selective covalent aldo-keto reductase family 1 member C3 (AKR1C3) inhibitor with an IC50 value of 13 nM. RJG-2051 interferes with the metabolic process of substrates such as androgens, estrogens, and prostaglandins by AKR1C3. RJG-2051 is promising for research of cancers[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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RJG-2051 | 99.42% | RJG-2051 is a selective covalent aldo-keto reductase family 1 member C3 (AKR1C3) inhibitor with an IC50 value of 13 nM. RJG-2051 interferes with the metabolic process of substrates such as androgens, estrogens, and prostaglandins by AKR1C3. RJG-2051 is promising for research of cancers. | ||||||||||||||||||||
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