3016437-05-8
3016437-05-8
Chemical Structure
Androgen receptor-IN-6
- CAS No.: 3016437-05-8
- Formula:C16H15N3OS
- Molecular Weight:297.37
InChIKey: LAJCSSWPGDDWCX-UHFFFAOYSA-N
SMILES: CN1C2=CC=C(C3=CC(C(N)=O)=CC=C3SC)C=C2C=N1
Biological Activity: Androgen receptor-IN-6 (compound 16) is an orally available androgen receptor (Androgen Receptor) potent inhibitor (IC50=0.12 μM in vitro), targeting the disordered N-terminal domain (NTD). Androgen receptor-IN-6 has good Caco2 cell membrane permeability and has an oral activity (F/%) of 16% in male CD-1 mice[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Androgen receptor-IN-6 | 98.07% | Androgen receptor-IN-6 (compound 16) is an orally available androgen receptor (Androgen Receptor) potent inhibitor (IC50=0.12 μM in vitro), targeting the disordered N-terminal domain (NTD). Androgen receptor-IN-6 has good Caco2 cell membrane permeability and has an oral activity (F/%) of 16% in male CD-1 mice. | ||||||||||||||||||||
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