3032600-19-1
Chemical Structure
CSD-CH2(1,8)-NH2
- CAS No.: 3032600-19-1
- Formula:C76H125N25O15S2
- Molecular Weight:1693.09
InChIKey: KUPKENZACMICGA-HAQFKNNNSA-N
SMILES: O=C(N[C@H](C(NCC(NCC(N[C@@H](CC1=CC=CC=C1)C(N[C@@H](CC(C)C)C(N[C@H]2CCCNC(N)=N)=O)=O)=O)=O)=O)CC3=CC=C(C=C3)O)CCSCSC[C@@H](C(N[C@H](C(N4CCC[C@H]4C(N[C@H](C(N[C@@H](CC(C)C)C(N[C@H](C(N)=O)CCCCN)=O)=O)CCCCN)=O)=O)CCCNC(N)=N)=O)NC([C@@H](NC2=O)CCCNC(N)=N)=O
Biological Activity: CSD-CH2(1,8)-NH2 is a selective and competitive KOR antagonist (Ki: 6.8 nM). CSD-CH2(1,8)-NH2 inhibits calcium mobilization in DRG neurons. CH2(1,8)-NH2 antagonizes the antinociceptive effect of U50,488. CSD-CH2(1,8)-NH2 can be used for research of neuropsychiatric disorders[1].
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CSD-CH2(1,8)-NH2 | CSD-CH2(1,8)-NH2 is a selective and competitive KOR antagonist (Ki: 6.8 nM). CSD-CH2(1,8)-NH2 inhibits calcium mobilization in DRG neurons. CH2(1,8)-NH2 antagonizes the antinociceptive effect of U50,488. CSD-CH2(1,8)-NH2 can be used for research of neuropsychiatric disorders. | |||||||||||||||||||||
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