3038478-21-3
Chemical Structure
MC4R antagonist-2
- CAS No.: 3038478-21-3
- Formula:C26H29F3N6O3
- Molecular Weight:530.55
IUPAC Name: (R)-1-((S)-7-((5-(2-(difluoromethoxy)-1-methyl-1H-imidazol-4-yl)-6-methylpyridin-2-yl)amino)-5-azaspiro[2.4]heptan-5-yl)-2-(5-fluoro-2-methoxypyridin-4-yl)propan-1-one
InChIKey: YMDSWECYBZOSSE-JLTOFOAXSA-N
SMILES: N([C@H]1C2(CN(C([C@H](C)C=3C=C(OC)N=CC3F)=O)C1)CC2)C=4N=C(C)C(=CC4)C=5N=C(OC(F)F)N(C)C5
Biological Activity: MC4R antagonist-2 is a potent melanocortin 4 receptor (MC4R) antagonist with an IC50 of 0.54 nM. MC4R antagonist-2 can be used for the research of MC4R-mediated conditions, such as cachexia, osteoporosis, neuropathic pain, depression, hypertension, malnutrition-related obesity, and associated inflammatory diseases[1].
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MC4R antagonist-2 | MC4R antagonist-2 is a potent melanocortin 4 receptor (MC4R) antagonist with an IC50 of 0.54 nM. MC4R antagonist-2 can be used for the research of MC4R-mediated conditions, such as cachexia, osteoporosis, neuropathic pain, depression, hypertension, malnutrition-related obesity, and associated inflammatory diseases. | |||||||||||||||||||||
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