3052544-42-7
3052544-42-7
Chemical Structure
GRPR antagonist-2
- CAS No.: 3052544-42-7
- Formula:C28H32F3N5O4
- Molecular Weight:559.58
IUPAC Name: tert-butyl 4-(((4-(trifluoromethyl)phenyl)carbamoyl)-L-tryptophyl)piperazine-1-carboxylate
InChIKey: WTVXQEPXYFGAJP-QHCPKHFHSA-N
SMILES: CC(C)(OC(N1CCN(CC1)C([C@H](CC2=CNC3=C2C=CC=C3)NC(NC4=CC=C(C=C4)C(F)(F)F)=O)=O)=O)C
Biological Activity: GRPR antagonist-2 is a potent gastrin releasing peptide receptor (GRPR) antagonist, having the cytotoxicity against certain cancer cells (IC50 of 0.77 and 2.5 μM in HGC-27 and Pan02 cells, respectively). Anticancer activity[1].
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GRPR antagonist-2 | GRPR antagonist-2 is a potent gastrin releasing peptide receptor (GRPR) antagonist, having the cytotoxicity against certain cancer cells (IC50 of 0.77 and 2.5 μM in HGC-27 and Pan02 cells, respectively). Anticancer activity. | |||||||||||||||||||||
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