3052930-88-5
3052930-88-5
Chemical Structure
Cathepsin L/S-IN-1
- CAS No.: 3052930-88-5
- Formula:C29H33BrN4O4S
- Molecular Weight:613.57
IUPAC Name: methyl N6-(bicyclo[2.2.1]heptan-2-yl)-N2-(4-(tert-butyl)benzoyl)-L-phenylalanyl-L-alanyl-L-leucyl-N6-methyl-L-lysyl-L-serinate 2,2,2-trifluoroacetate
InChIKey: QSUSOTUHCHGTAN-KAYWLYCHSA-N
SMILES: O[C@@H](COC[C@H](NS(=O)(C1=CC=C(C=C1)Br)=O)CC2=CC=CC=C2)CN(CC3)CCN3C(C=CC=C4)=C4C#N
Biological Activity: Cathepsin L/S-IN-1 is a dual inhibitor of Cathepsin L and Cathepsin S with IC50s of 4.10 μM and 1.79 μM, respectively. Cathepsin L/S-IN-1 shows a significant antimetastatic and invasive effects on pancreatic cancer BxPC-3 and PANC-1 cells[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Cathepsin L/S-IN-1 | 99.89% | Cathepsin L/S-IN-1 is a dual inhibitor of Cathepsin L and Cathepsin S with IC50s of 4.10 μM and 1.79 μM, respectively. Cathepsin L/S-IN-1 shows a significant antimetastatic and invasive effects on pancreatic cancer BxPC-3 and PANC-1 cells. | ||||||||||||||||||||
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